@article{3ae8099d1ce34bfaba56ca4ba5d6ef1f,
title = "Synthesis, biological evaluation and radiolabelling by 18F- fluoroarylation of a dopamine D3-selective ligand as prospective imaging probe for PET",
abstract = "Radical 18F-fluoroarylation with fluorine-18-labelled arenediazonium chlorides has been successfully applied to the radiochemical synthesis of the dopamine D3-selective ligand SH 317 ([ 18F]8). SH 317 has been evaluated as a new PET ligand candidate by in vivo experiments.",
keywords = "18-Fluorine, Dopamine, Ligands, Positron emission tomography, Radiochemical labelling",
author = "H{\"o}fling, {S. B.} and S. Maschauer and H. H{\"u}bner and P. Gmeiner and Wester, {H. J.} and O. Prante and Heinrich, {M. R.}",
note = "Funding Information: The authors would like to thank the Friedrich-Alexander-Universit{\"a}t Erlangen-N{\"u}rnberg (FAU) and the Deutsche Forschungsgemeinschaft (DFG) [DFG ( HE5413/3-1 ), DFG ( WE 2386/5-1 ), DFG ( PR 677/2-3 )] for generous financial support. ",
year = "2010",
month = dec,
day = "1",
doi = "10.1016/j.bmcl.2010.09.142",
language = "English",
volume = "20",
pages = "6933--6937",
journal = "Bioorganic and Medicinal Chemistry Letters",
issn = "0960-894X",
publisher = "Elsevier Ltd.",
number = "23",
}