Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles

Julian Wippich; Ingo Schnapperelle; Thorsten Bach

doi:10.1039/c4cc10144h

Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles

Julian Wippich
, Ingo Schnapperelle
, Thorsten Bach

Lehrstuhl für Organische Chemie I

Technische Universität München

Publikation: Beitrag in Fachzeitschrift › Artikel › Begutachtung

35 Zitate (Scopus)

Abstract

A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag₂CO₃ and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.

Originalsprache	Englisch
Seiten (von - bis)	3166-3168
Seitenumfang	3
Fachzeitschrift	Chemical Communications
Jahrgang	51
Ausgabenummer	15
DOIs	https://doi.org/10.1039/c4cc10144h
Publikationsstatus	Veröffentlicht - 21 Feb. 2015

Zugriff auf Dokument

10.1039/c4cc10144h

Andere Dateien und Links

Verknüpfung zur Publikation in Scopus

Dieses zitieren

@article{977016685e354241a1910bc924039558,

title = "Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles",

abstract = "A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99\% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag2CO3 and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.",

author = "Julian Wippich and Ingo Schnapperelle and Thorsten Bach",

note = "Publisher Copyright: {\textcopyright} The Royal Society of Chemistry 2015.",

year = "2015",

month = feb,

day = "21",

doi = "10.1039/c4cc10144h",

language = "English",

volume = "51",

pages = "3166--3168",

journal = "Chemical Communications",

issn = "1359-7345",

publisher = "Royal Society of Chemistry",

number = "15",

}

TY - JOUR

T1 - Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles

AU - Wippich, Julian

AU - Schnapperelle, Ingo

AU - Bach, Thorsten

PY - 2015/2/21

Y1 - 2015/2/21

N2 - A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag2CO3 and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.

AB - A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag2CO3 and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.

UR - https://www.scopus.com/pages/publications/84929997044

U2 - 10.1039/c4cc10144h

DO - 10.1039/c4cc10144h

M3 - Article

AN - SCOPUS:84929997044

SN - 1359-7345

VL - 51

SP - 3166

EP - 3168

JO - Chemical Communications

JF - Chemical Communications

IS - 15

ER -

Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles

Abstract

Zugriff auf Dokument

Andere Dateien und Links

Fingerprint

Dieses zitieren