Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles

Julian Wippich; Ingo Schnapperelle; Thorsten Bach

doi:10.1039/c4cc10144h

Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles

Julian Wippich, Ingo Schnapperelle, Thorsten Bach

Lehrstuhl für Organische Chemie I

Technische Universität München

Publikation: Beitrag in Fachzeitschrift › Artikel › Begutachtung

34 Zitate (Scopus)

Abstract

A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag₂CO₃ and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.

Originalsprache	Englisch
Seiten (von - bis)	3166-3168
Seitenumfang	3
Fachzeitschrift	Chemical Communications
Jahrgang	51
Ausgabenummer	15
DOIs	https://doi.org/10.1039/c4cc10144h
Publikationsstatus	Veröffentlicht - 21 Feb. 2015

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title = "Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles",

abstract = "A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag2CO3 and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.",

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doi = "10.1039/c4cc10144h",

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T1 - Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles

AU - Wippich, Julian

AU - Schnapperelle, Ingo

AU - Bach, Thorsten

PY - 2015/2/21

Y1 - 2015/2/21

N2 - A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag2CO3 and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.

AB - A total of 19 alkylated heterocycles (thiophenes, benzothiophenes, pyrroles, furans) were prepared (36-99% yield) from the respective pyridin-2-yl-substituted precursors employing alkylboronic acids as the C-H alkylating reagents in an oxidative (Ag2CO3 and 2,6-dimethyl-1,4-benzoquinone as oxidants) Pd-catalysed coupling reaction.

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U2 - 10.1039/c4cc10144h

DO - 10.1039/c4cc10144h

M3 - Article

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VL - 51

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JO - Chemical Communications

JF - Chemical Communications

IS - 15

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Regioselective oxidative Pd-catalysed coupling of alkylboronic acids with pyridin-2-yl-substituted heterocycles

Abstract

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